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Cheng Chen†, Zhengwei Ding†, Yan Gao†, Yi Jing†, Yong-An Luo†, Xingxing Ma†, Xuenian Chen*, Pengfei Li*, Zaozao Qiu*, Qiuling Song*, Xiao-Ye Wang*, Zuowei Xie*
Sci. China Chem., 2025, 68, DOI: 10.1007/s11426-025-2886-2.
Shanghui Tian, Ruxue Liu, Kuan Zhang, Yan Xia, Yinuo Liu, Pengfei Li, Xin-Hua Duan,* Li-Na Guo*
Org. Lett. 2025, 27, 3818.
Kuan Zhang, Zhengyang Gao, Yan Xia, Pengfei Li, Pin Gao, Xin-Hua Duan, Li-Na Guo*
Chem. Sci., 2025, 16, 1411.

Lulu Qin, Tao Yu, Zhengwei Ding, Min Zhao, Pengfei Li*
Synthesis, 2025, 57, DOI: 10.1055/a-2511-4274.

Tao Yu, Xue Zhao, Zaicheng Nie, Lulu Qin, Zhengwei Ding, Liang Xu, Pengfei Li*
Angew. Chem. Int. Ed. 2025, e202420831

Kuan Zhang, Yan Xia, Shanghui Tian, Xin-Hua Duan, Pengfei Li,* Li-Na Guo*
ChemCatChem 2025, e202401909

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88. Pyridine-boryl radical-catalyzed [3p + 2s] cycloaddition for the synthesis of pyridine isosteres
Yuan Liu, Shuang Lin, Zhengwei Ding, Yin Li, Ya-Jie Tang, Jiang-Hao Xue, Qingjiang Li, Pengfei Li,* Honggen Wang*
Chem 2024, DOI: 10.1016/j.chempr.2024.08.010

87. Regio- and Diastereoselective Synthesis of Polysubstituted Piperidines Enabled by Boronyl Radical-Catalyzed (4+2) Cycloaddition
Zhengwei Ding, Zhijun Wang, Yingying Wang, Xicheng Wang, Yuanji Xue, Ming Xu, Hailong Zhang,* Liang Xu, * Pengfei Li*
Angew. Chem. Int. Ed. 2024, 63, e202406612

86. Broad-Scope (3+2) Cycloaddition of Cyclopropanes and Alkynes Enabled by Boronyl Radical Catalysis
Jingru Wen#, Zhengwei Ding#*, Pengfei Li*
Org. Lett. 2024, 26, 7021.

85. Vinylcyclopropane-Cyclopentene (VCP-CP) Rearrangement Enabled by Pyridine-Assisted Boronyl Radical Catalysis
Ting Li, Lanfeng Wei, Zhijun Wang, Xinyu Zhang, Jinbo Yang, Yu Wei,* Pengfei Li,* Liang Xu*
Org. Lett. 2024, 26, 5341.
84. Lewis Acid-Catalyzed Formal [2π+2σ] Cycloaddition of Bicyclobutanes with Quinoxalin-2(1H)-ones: Access to Quinoxaline-Fused Aza-Bicyclo[2.1.1]hexanes
Kuan Zhang, Shanghui Tian, Wenke Li, Xu Yang, Xin-Hua Duan, Li-Na Guo,* Pengfei Li*
Org. Lett. 2024, 26, 5482.
83. Asymmetric Total Synthesis of Pedrolide (Highlight)
Ruiqi Si, Pengfei Li*
Chin. J. Org. Chem. 2024, 44, 1031.
82. Design and Application of New Pyridine-Derived Chiral Ligands in Asymmetric Catalysis
Shuai Zhang, Yizhao Ouyang, Yuan Gao, Pengfei Li*
Acc. Chem. Res. 2024, 57, 957.
81. Chemoenzymatic β-Specific Methylene C(sp3)–H Deuteration of Carboxylic Acid
Xicheng Wang,# Zhaohui Sun,# Tao Li,# Saima Perveen, Pengfei Li* (#co-first author)
Green Chem. 2024, 26, DOI: 10.1039/D4GC00082J.
80. Iridium-Catalyzed Doubly Stereoconvergent Allylic Alkylation of Racemic α-Boryl Organozinc Reagents
Jinhui Han, Xirong Liu, Hao Jin, Panchi Guo, Liang Xu, Pengfei Li,* Miao Zhan*
Chem Catal. 2024, 4, DOI: 10.1016/j.checat.2023.100858.

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79. Synthesis of Isoquinoline-3-carboxylate Chelated B,B-Diaryl Tetracoordinated Organoboron Complexes
Weina Tian, Liang Xu, Yu Wei,* Pengfei Li*
Chin. J. Org. Chem. 2023, 43, 1792.

78. Visible Light-Mediated Organoboron-Catalyzed Metal-Free Synthesis of Silanols from Silanes
Jinbo Yang, Xiangxue Cao, Lanfeng Wei, Jianshu Zhan, Jinli Zhang, Ping Liu, Liang Xu,* Pengfei Li
Molecules 2023, 28, 4082.
77. Asymmetric Synthesis of Metallacarboranes using a Traceless Chiral Auxiliary
Jiao Jiao, Pei He, Tilong Yang, Tingwei Zhang, Linghua Wang, Tian Han, Yong Nie, Zhenyang Lin, Pengfei Li*
Org. Chem. Front., 2023, 10, 5965.
76. Additive-Free Transfer Hydrogenative Direct Asymmetric Reductive Amination Using a Chiral Pyridine-Derived Half-Sandwich Catalyst
Yuan Gao, Zhijun Wang, Xinyu Zhang, Min Zhao, Shuai Zhang, Chao Wang, Liang Xu,* Pengfei Li*
Angew. Chem. Int. Ed. 2023, 62, e202303709.

Panchi Guo, Hao Jin, Jinhui Han, Liang Xu, Pengfei Li*, Miao Zhan*
Org. Lett. 2023, 25, 1268.

Tao Yu, Jinbo Yang, Zhijun Wang, Zhengwei Ding, Ming Xu, Jingru Wen, Liang Xu, Pengfei Li*
J. Am. Chem. Soc. 2023, 145, 4304.

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Ming Xu, Zhijun Wang, Zhaohui Sun, Yizhao Ouyang, Zhengwei Ding, Tao Yu, Liang Xu, Pengfei Li*
Angew. Chem. Int. Ed. 2022, 61, e202214507.
Hot Paper

Linghua Wang, Tao Li, Saima Perveen, Shuai Zhang, Xicheng Wang, Yizhao Ouyang, Pengfei Li*
Angew. Chem. Int. Ed. 2022, 61, e202213943.

Saima Perveen,# Shuai Zhang,# Linghua Wang, Peidong Song, Yizhao Ouyang, Jiao Jiao, Xin-Hua Duan, Pengfei Li* (# co-first author)
Angew. Chem. Int. Ed. 2022, 61, e202212108.

Shuai Mao,*# Bo Yuan,# Xinyu Wang, Yahao Zhao, Lu Wang, Xue-Yan Yang, Yi-Ming Chen, San-Qi Zhang,* Pengfei Li* (# co-first author)
Org. Lett. 2022, 24, 3594.
69. Catalysis with Diboron(4)/Pyridine: Application to the Broad-Scope [3+2] Cycloaddition of Cyclopropanes and AlkenesZhengwei Ding,# Zhi Liu,# Zhijun Wang, Tao Yu, Ming Xu, Jingru Wen, Kaiyan Yang, Hailong Zhang, Liang Xu,* Pengfei Li* (# co-first author)
J. Am. Chem. Soc. 2022, 144, 8870.
Featured in Org. Chem. Highlights

Ming Xu, Yizhao Ouyang, Linghua Wang, Shuai Zhang, Pengfei Li*
Chem. Commun. 2022, 58, 3677.

Shuai Zhang,# Saima Perveen,# Yizhao Ouyang,# Liang Xu, Tao Yu, Min Zhao, Linghua Wang, Peidong Song, Pengfei Li*(# co-first author)
Angew. Chem. Int. Ed. 2022, 61, e202117843.
Hot Paper
Wiley | Top Dowloaded Author(Wiley年度高下载量作者奖)

Tengfei Ma, Xinyun Zhai,* Yongkang Huang, Mengzhen Zhang, Pengfei Li, Yaping Du
J. Rare Earths. 2022, 40, 1407.

Yu Liu, Miao Zhan,* Pengfei Li*
Chin. J. Chem. 2022, 40, 1028

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Siyi Ding, Huaping Ren, Min Zhu, Qiang Ma, Zongcheng Miao,* Pengfei Li*
Synth. Commun. 2020, 51, 593.

Jiao Jiao,* Wenzheng Nie, Tao Yu, Fan Yang, Qian Zhang, Feierdaiweisi Aihemaiti, Tingjun Yang, Xuanyu Liu, Jiachen Wang, Pengfei Li*
Chem. Eur. J. 2020, 26, 4817.

Zhengwei Ding, Zhi Liu, Guanghu Tong, Linlin Hu, Yangqing He,* Yueyun Bao, Zhouhang Lei, Hailong Zhang, Pengfei Li*
Org. Chem. Front. 2020, 7, 1862.

Guanghu Tong, Zhengwei Ding, Zhi Liu, You-Song Ding, Liang Xu,* Hailong Zhang, Pengfei Li*
J. Org. Chem. 2020, 85, 4813.

Miao Zhan, Peidong Song, Jiao Jiao, Pengfei Li*
Chin. J. Chem. 2020, 38, 665.

Miao Zhan, Zhengwei Ding, Shaozhi Du, Haohua Chen, Chao Feng, Ming Xu, Zhi Liu, Mengxi Zhang, Chao Wu, Yu Lan,* Pengfei Li*
Nat. Commun. 2020, 11, 792.

康强,曹晓宇, 刘磊, 李鹏飞, 吴长征,杨鹏,崔琳,陈拥军
中国科学基金
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Tao Yu, Zhengwei Ding, Wenzheng Nie,Jiao Jiao,* Hailong Zhang, Qian Zhang, Chao Xue, Xinhua Duan, Yoichi M. A. Yamada, Pengfei Li*
Chem. Eur. J. 2019, 26, 5729.

Xiaodong Yang, Bingjie Zhang, Sikun Zhang, Guoping Li, Letian Xu, Zhijun Wang, Pengfei Li, Yanfeng Zhang, Zishun Liu, Gang He*
Org. Lett. 2019, 21, 8285.
Cover paper

Jun-Cheng Yang, Lei Chen, Fan Yang, Pengfei Li, Li-Na Guo*
Org. Chem. Front. 2019, 6, 2932.

Xiaoying Xu, Qian Zhang, * Kang Liu, Nailiang Liu, Ying Han,* Weixing Chen, Chao Xie, Pengfei Li, Jie He*
Polym. Chem. 2019, 10, 3585.
Back cover article
Yizhao Ouyang, Miao Zhan, Jing Zhou,Jiao Jiao, Hao Hu, Yoichi M. A. Yamada,* Pengfei Li*
Chin. J. Chem. 2019, 37, 807.
Siyi Ding, Linghua Wang, Zongcheng Miao,* Pengfei Li*
Molecules 2019, 24, 1434.

Shuai Mao, Zhengkai Chen, Lu Wang, Daulat Bikram Khadka, Minhang Xin, Pengfei Li,* San-Qi Zhang*
J. Org. Chem. 2019, 84, 463.

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Guanghu Tong, Zhi Liu, Pengfei Li,*
Chem 2018, 12, 2944.

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Li Liu, Guanghui Wang, Jiao Jiao, Pengfei Li*
Org. Lett. 2017, 19, 6132.

Liang Xu, Guanghui Wang, Shuai Zhang, Hong Wang, Linghua Wang, Li Liu, Jiao Jiao, Pengfei Li*
Tetrahedron 2017, 73, 7123.

Hong Wang, Guanghui Wang, Pengfei Li*
Org. Chem. Front. 2017, 4, 1943.

Kai Chen, Linghua Wang, Ge Meng,* Pengfei Li*
Synthesis 2017, 49, 4719.

Dawei Hu, Linghua Wang, Pengfei Li*
Org. Lett. 2017, 19, 2770.

Chao Wu, Xiufang Hou, Yuheng Zheng, Pengfei Li, Dongmei Lu*
J. Org. Chem. 2017, 82, 2898.
Qian Zhang,* Shuhuan Yang, Tingting Zhu, Jung Kwon Oh, Pengfei Li
React. Funct. Polym. 2017, 110, 30.
Guanghui Wang, Li Liu, Hong Wang, You-Song Ding, Jing Zhou, Shuai Mao, Pengfei Li*
J. Am. Chem. Soc. 2017,139, 91.

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Xiaojuan Zhang, Qian Zhang,* Yuzhen Wu, Chao Feng, Chao Xie, Xiaodong Fan, Pengfei Li
Macromol. Rapid. Commun. 2016, 37, 1311.
Cover Article

Kai Chen, Man Sing Cheung, Zhenyang Lin,* Pengfei Li*
Org. Chem. Front. 2016, 3, 875.
Hot paper

Kai Chen, Pei He, Shuai Zhang, Pengfei Li*
Chem. Commun. 2016, 52, 9125.

Kai Chen, Shuai Zhang, Pei He, Pengfei Li*
Chem. Sci. 2016, 7, 3676.

Siyi Ding, Liang Xu, Pengfei Li*
ACS Catal. 2016, 6, 1329.

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Xiaojuan Zhang, Qian Zhang,* Chao Xie, Aiting Gao, Zheng Chang, Jung Kwon Oh, Peng Yang, Pengfei Li*
J. Polymer Sci. Part A: Polymer Chem. 2015, 54, 1396.
Yue Wang, Qian Zhang,* Chao Xie, Xin Zhao, Jinfen Niu, Jie Zhao, Jung Kwon Oh, Peng Li, Pengfei Li*
RSC Adv. 2015, 5, 95666.
Liang Xu, Shuai Zhang, Pengfei Li*
Chem. Soc. Rev. 2015, 44, 8765.
Guanghui Wang,† Liang Xu,† Pengfei Li* († These authors contributed equally.)
J. Am. Chem. Soc. 2015, 137, 8058.

Chao Feng, Hong Wang, Liang Xu, Pengfei Li*
Org. Biomol. Chem. 2015, 26, 7136.

Liang Xu†, Shuai Zhang†, Pengfei Li* († These authors contributed equally.)
Org. Chem. Front. 2015, 2, 459.
Inside front cover article

Liang Xu, Pengfei Li*
Chem. Commun. 2015, 51, 5656.

Zhengzheng Chen, Pengfei Li,* Chao Wu*
RSC Adv. 2015, 5, 11791.
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Liang Xu, Pengfei Li*
Synlett 2014, 25, 1799.
Invited SYNPACTS.

Guanghu Tong, Zhi Liu, Pengfei Li*
Org. Lett. 2014, 16, 2288.

Dongmei Lu,* Chao Wu, Pengfei Li*
Org. Lett. 2014, 16, 1486.
Liang Xu,† Siyi Ding,† Pengfei Li* (†These authors contributed equally.)
Angew. Chem. Int. Ed. 2014, 53, 1822.
Highlighted by Synlett 2014, 1799.
Highlighted by Chinese J. Org. Chem. 2014, 34, 836.

Dongmei Lu,* Chao Wu, Pengfei Li*
Chem. Eur. J. 2014, 20, 1630.

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Xiaowu Liu, Fei Xiong, Xuanping Huang, Liang Xu, Pengfei Li,* Xiaoxing Wu,*
Angew. Chem. Int. Ed. 2013, 52, 6962
Highlighted by Synlett, 2013, 24, 1882.
Highlighted by Chinese J. Org. Chem. 2013, 33, 1850.

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Patents
6. 一种手性稠环[6-5-3]吡啶二醇的合成方法
李鹏飞; 王西城; 杨婧; 张帅; 张乾
CN202311068689.7
6. 一种手性2,2’-联吡啶配体及其制备方法和应用
李鹏飞; 欧阳彝钊; 张帅; 茜姆勃玟; 宋沛东
CN202111434132.1
5. 手性吡啶衍生的N,B配体及制备方法和在铱催化不对称硼化反应中的应用
李鹏飞; 宋沛东
CN202011602455.2
4. 一种硫代硅烷配体及其制备方法和在芳基硼化催化反应中的应用
李鹏飞; 聂文政; 宋沛东
CN201911150320.4
3. 一种手性2,2’-联吡啶配体及其制备方法和在制备手性环丙烷衍生物中的应用
李鹏飞; 欧阳彝钊; 占苗
CN201910394448.9
2. 一种巴豆烷二萜Prostratin的化学全合成制备方法
李鹏飞; 佟广虎
CN201810307255.0
1. 硼烷吡啶前配体及其制备方法和应用以及制备芳基硼酸酯的方法
李鹏飞; 王光辉; 徐亮
CN201510067478.0
Book Chapters
1. "Di- and Polyboron Compounds: Preparation and Chemoselective Transformations” in Boron reagents in synthesis (Edited by Adiel Coca)
Liang Xu, Shuai Zhang, Pengfei Li
American Chemical Society, 2016
2. “New Design of Phenol-containing Polymers as Radical Scavengers” in Free Radicals and Health (Edited by Marianne Rutherford)
Qian Zhang, Yunyue Jiang, Yue Wang, Peng Li, Xin Zhao, Chao Xie, Jie Zhao, Jinfen Niu, Jung Kwon Oh, Pengfei Li
Nova Science Publishers, 2016
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15. A Microfluidic System for the Continuous Recycling of Unmodified Homogeneous Palladium Catalysts via Liquid-Liquid Phase Separation
Pengfei Li,* Jason S. Moore, Klavs F. Jensen*
ChemCatChem 2013, 5, 1729
14. Modular Total Synthesis of Rhizopodin: A Highly Potent G-Actin Dimerizing Macrolide
Manuel Kretschmer, Michael Dieckmann, Pengfei Li, Sven Rudolph, Daniel Herkommer, Johannes Troendlin, Dirk Menche,*
Chem. Eur. J. 2013, 19, 15993
13. Total Synthesis of Rhizopodin
Michael Dieckmann, Manuel Kretschmer, Pengfei Li, Sven Rudolph, Daniel Herkommer, Dirk Menche
Angew. Chem. Int. Ed. 2012, 51, 5667
12. Continuous-Flow Synthesis of 3,3-Disubstituted Oxindoles by a Palladium-Catalyzed a-Arylation/Alkylation Sequence
Pengfei Li, Stephen L. Buchwald*
Angew. Chem. Int. Ed. 2011, 50, 6396
11. Concise Synthesis of Tetrahydropyrans by a Tandem Oxa-Michael/Tsuji-Trost Reaction
Liang Wang, Pengfei Li, Dirk Menche*
Angew. Chem. Int. Ed. 2010, 49, 9270
10. Stereoselective Total Synthesis of Etnangien and Etnangien Methyl Ester
Pengfei Li, Jun Li, Fatih Arikan, Wiebke Ahlbrecht, Michael Dieckmann, Dirk Menche*
J. Org. Chem. 2010, 75, 2429
9. Stereodivergent Synthesis of 1,3-syn- and anti-Tetrahydropyrimidinones
Michael Morgen, Sebastian Bretzke, Pengfei Li, Dirk Menche*
Org.Lett. 2010, 12, 4494
8. Design, Synthesis and Biological Evaluation of Simplified Analogues of the RNA Polymerase Inhibitor Etnangien
Dirk Menche*, Pengfei Li, Herbert Irschik
Bioorg. Med. Chem. Lett. 2010, 20, 939
7. Total Synthesi of Etnangien
Pengfei Li, Jun Li, Fatih Arikan, Wiebke Ahlbrecht, Michael Dieckmann, Dirk Menche*
J. Am. Chem. Soc. 2009, 131, 11678
6. An Efficient Procedure for the Direct Nucleophilic Substitution of the Abiko-Masamune Auxiliary
Jun Li, Pengfei Li, Dirk Menche*
Synlett 2009, 2417
5. Cycloadditions in the Total Synthesis of Sporolide B
Pengfei Li, Dirk Menche*Angew. Chem. Int. Ed. 2009, 48, 50784. Synthesis and Characterization of New 4-(Substituted pyrimidin-2-yl)-1-(Substituted benzensulfonyl)- semicarbazides
Pengfei Li, Bao-Lei Wang, Ning Ma, Su-Hua Wang, Zheng-Ming Li*
Chin. J. Org. Chem. 2005, 25, 1057
3. Synthesis and Herbicidal Activity of New Sulfonylurea Derivatives
Pengfei Li, Ning Ma, Bao-Lei Wang, Zheng-Ming Li*, Su-Hua Wang, Yong-Hong Li
Chem. J. Chinese Uni. 2005, 26, 1459
2. Synthesis of 2-Chlorosulfonylbenzoyl Chloride,
Pengfei Li, Bao-Lei Wang, Ning Ma, Zheng-Ming Li*, Su-Hua Wang
Chemical Reagents 2005, 27, 445
1. Synthesis and Biological Activity of New Phenylsulfonylurea Derivatives
Ning Ma, Pengfei Li, Yong-Hong Li, Zheng-Ming Li*, Ling-Xiu Wang, Su-Hua Wang
Chem. J. Chinese Uni. 2004, 25, 2259






